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Buy 99% Tianeptine Sodium Powder In Stock

Why You Should Buy Tianeptine Powder From Us?

#1. SAFE SHIPPING!!!:

WE HAVE ABLE COURIER AGENT TO MAKE YOU GET IT SAFELY&QUICKLY.

#2. High quality standards with the best price you can ever find in the market. (EP9.0 and MOQ starts at 100G)

#3. Quality guarantee: 100% refund for any quality issues after testing.

#4. Fast shipment: goods will be shipped out after rapid repacking and tracking number will be provided to you within 3~4 days.

#5. Steady supply: we keep kilos in stock for prompt shipment. Repacking can be arranged within 1 working day!

Looking For Tianeptine Sodium Vendors? Contact Us Now!

What Is Tianeptine Sodium?

Tianeptine sodium structure

Cas number: 30123-17-2

Molecular Formula: C21H24ClN2NaO4S

Molecular Weight: 458.9 g/mol

HS Code: 2934991000

Pure Tianeptine sodium is a white to yellowish and very hygroscopic powder.

The color difference is partially caused by water content inside or by impurity.

When its purity is over 99%, it tends to be white rather than yellowish.

As it is stronly prone to absorb moistures in the air, it should be sealed and stored properly before they become rocks after leeching water.

It has been used as an atypical antidepressant for the treatment of the major depressive disorders. It is also used to treat anxiety, asthma, and irritable bowel syndrome.

It is one of our most competitive pharmaceutical ingredients in stock. It is marketed as Stablon and Coaxil in many countries.

Peolple also use it for treating pain caused by fibromyalgia because of its anticonvulsant and analgesic effects. It has been effective in the treatment of attention-deficit hyperactivity disorder with minimal side effects too.

Is Tianeptine Sodium A Nootropic?

The answer is Yes.

Nootropics, also known as smart drugs, are used to improve cognitive function, particularly executive functions, memory, creativity, or motivation in healthy individuals.

Tianeptine is a TCA-like and serotonergic enhancing medication prescribed commonly in the Middle East and Europe for depression and anxiety.

However, the study shows it does help to improve people’s cognitive functions.

The FDA has not approved Tianeptine for any use in the United States for any conditions, let alone allow it to be used to improve cognitive functions.

Tianeptine Sodium vs Sulfate

Tianeptine sodium vs sulfate

There are three commonly seen Tianeptine forms on the market: Tianeptine free acid, sodium salt, and tianeptine sulfate salt.

Among them, tianeptine acid is the least popular and cheapest type.

Maybe tianeptine free acid only exists because it can be made into various tianeptine salts such as tianeptine hydrochloride, tianeptine tosylate, tianeptine phosphate, etc.

So here we only list the difference between tianeptine sodium and tianeptine sulfate (also written as tianeptine sulphate). 

1. Their age. (Sodium is older than sulfate)

Sodium tianeptine is the first to be widely used for medical purposes for depression since 1960.

Tianeptine sulfate is later developed and improved versions to replace the sodium form.

2. Stability. (sulfate salt is more stable than sodium salt)

Both tianeptine sodium and sulphate are stable when protected from light and air. But sodium salt is very hygroscopic to get chunky. While tianeptine sulfate salt contains monohydrate with itself, it is more stable when exposed to air for a short period.

3. Water solubility uniformity. (Tianeptine sulfate has better uniformity than sodium)

In water solutions PH ranged 1~6, the soluble amount of tianeptine sulphae in water is very average.

Its solubility curve is very smooth, the value gets slightly smaller as the PH goes up. While sodium salt has a sudden drop when PH goes from 1 to 6. As the stomach fluid PH ranges from 1.5~3.5 and sure you will choose sulphate to maintain a stable solubility.

4. Taste. (Tianeptine sulfate is not bitter, sodium is)

 The bitterness of sodium tianeptine can linger in your mouth for one month if it is taken directly.

While tianeptine sulphate is much better on the taste, no such strong bitterness at all.

That’s why you only see tianeptine sodium capsules but rarely see any tianeptine sodium tablets on the market.

5. Half-life and Bioavailability. (Tianeptine sulfate lasts longer than sodium)

According to researches and online reviews, tianeptine sulphate performs better on both half-life and bioavailability. Sulphate is easier to absorb and its effect lasts longer, while dosing sodium can go to 6~7 times daily to obtain the same effect as sulphate.

6. Price. (Tianeptine Sulfate is 20% higher than sodium)

As tianeptine sulfate has better performance almost on any aspect than tianeptine sodium and the production process is a little more complicated, its price is also a little higher, which does make sense.

Tianeptine vs Trazodone

Tianeptine sodium vs trazadone

Both Trazodone hcl and Tianeptine can be used for the treatment of depression.

What are their differences?

#1. Different Indications.

Tianeptine sodium is mainly used for the treatment of classic depressive episodes.

Trazodone is a tetracyclic atypical antidepressant that selectively antagonizes 5-hydroxytryptamine (5-HT) reuptake and weakly blocks norepinephrine (NA) reuptake, but has no effect on dopamine (DA), histamine or acetylcholine.

It will not inhibit the activity of monoamine oxidase inhibitors (MAO) in the brain.

In addition, trazodone has antagonistic effects on 5-HT2A receptors or 5-HT2C receptors.

Trazadone can improve sleep, significantly shorten the sleep latency of depressed patients, prolong the overall sleep time and improve sleep quality.

#2. Approval date and Range

Trazodone has been approved for medical use in the United States in 1981. It is used more widely.

It was approved in the Netherlands in 2014 in forms of 100mg tablets.

While Tianeptine has not been authorized by USFDA for any indications in the United States until today.

Though tianeptine is approved and marketed in many European countries, the UK has not approved it yet for depression yet.

#3. Cost differences

Price for Trazodone as bulk ingredient is much lower.

The cost of trazodone is about 1/7 of that of Tianeptine.

Trazodone costs about 600~800USD/kilo, while price for tianeptine per kilo is around 7000USD.

What are Tianeptine Sodium's Side Effects?

#1. Common side effects(>1% frequency)

Headache (up to 18%) / Dizziness (up to 10%) / Insomnia/nightmares (up to 20%) / Drowsiness (up to 10%) / Dry mouth (up to 20%) / Constipation (up to 15%) / Nausea  / Abdominal pain / Weight gain (~3%) / Agitation / Anxiety / irritability

#2. Uncommon side effects(0.1-1% frequency) 

Bitter taste / Flatulence / Gastralgia / Blurred vision / Muscle aches / Premature ventricular contractions / Micturition disturbances / Palpitations
Orthostatic hypotension / Hot flushes / Tremor Rare (<0.1% frequency) / Hepatitis / Hypomania / Euphoria / ECG changes / Pruritus / allergic-type / skin reactions / Protracted muscle aches

Warnings (tianeptine sodium withdrawal)

According to tianeptine marketer Servier, stopping of treatment with tianeptine is difficult, due to the possibility of withdrawal symptoms in a person. The severity of the tianeptine withdrawal is dependent on the daily dose, with high doses being extremely difficult to quit. DEA states that the withdrawal symptoms in humans typically result in agitation, nausea, vomiting, tachycardia, hypertension, diarrhea, tremor, and diaphoresis. 

Data are demonstrating that the abuse of tianeptine is increasing while contributing to the current opioid epidemic.

How Much Does Tianeptine Sodium Cost?

Currently we have it for sale and our running stock is 25kg to keep it always fresh.

The price from octagonchem for commercial order quantities of 50kg or more is around 2900USD/kg.

For quantities of 10kg, our cost is around 3000USD/KG.

If you only buy 1kilo, our price is about 3300USD/KG.

For costs of 100Gram, our offer is about 550USD including shipping.

As all prices are subject to the raw material price fluctuations, please contact us directly for more accurate prices.

For a better comparison, you check prices below from other online stores for your ref.

Price from tianeptinedirect is 6500usd per kilo

Tianeptinebuyonline is selling by 800usd per 100g

Price from tianeptinestore is 440usd per 50g

Cost from savant-research is 106usd per 10g

How Can You Buy Tianeptine Locally?

As you can see the prices from other suppliers above, their unit prices for 1kilo is over 7000USD as the wholesale price.

#1. If you are close to them and need them urgently, and you are willing to pay some extra dollars, so shipping from your local vendors means there won’t be need for your chemicals to pass borders. And you can choose them with lower MOQ to 10 Grams and Higher prices.

#2. If you are a buyer from another country other than the sellers are located, and they won’t ship the goods from your local warehouses, please contact us now for a quick order, we will manage to get you the best prices.

Currently we have 27.5 Kilo as Running Stock Ready For Fast Shipping.

You can check our terms below and prices from other suppliers above for your decision.

How Do You Ship and Store Bulk Tianeptine Sodium?

Firstly, let’s talk about the shipping options.

Tianeptine sodium is a safe chemical to be shipped by air or courier.

It is not dangerous or bio-poisonous, with RAT ORAL LD50 as over 1100mg/kilo.

It is not flammable or explosive, it can bear small bumps.

We’ve also get its certificate of safe air transportation from DGM, SRICI, etc, which is a firm proof for its safety as a common chemical.

If it is safe to be shipped by air or express, shipping by sea and rail won’t be a problem at all.

Secondly: For the storage and shipping conditions, we will break it one by one.

We have run stability tests for its storage, both at accelerated or common room temperature conditions. The stability tests have showed that it is stable for at least 24 months under room temperature, on the conditon of proper sealing and protection from the sunlight.

Though it is stable for 2 years by room temperature, it does not mean it will go bad during the transportation. You have to make sure thast the cabin temperature is not too high. Also you need to seal it well to protect it from possible moisture or light during the transportation.

When it has reached your warehouse, store it in a cool, dry and temperature-stable evironment.

Technical Documents Download

References

  1. Tianeptine in wikipedia
  2. Tianeptine In Pubchem
  3. https://www.drugbank.ca/salts/DBSALT001784
  4. https://patents.google.com/patent/US8198268B2/en
  5. https://www.quora.com/Whats-it-like-to-take-Tianeptine-sulfate
  6. Trazodone in wikipedia

Disclaimer

Our tianeptine series will not be sold to individuals, only to companies or institutions used for research only.

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